From: Tissue Inhibitor of Metalloproteinases-4. The road less traveled
TIMP-4 | Target MMP | Kinetic parameter | Key Residue(s) | Ref. |
---|---|---|---|---|
full-length | cdMMP-11 | K i 2.59 nM | ? | [57] |
full-lenght | cdMMP-11 | IC50 19 nM | ? | [55] |
full-lenght | MMP-1 | K i 0.65 nM | ? | [57] |
N-TIMP-42 | MMP-2 | K i app 0.3 nM | ? | [33] |
full-lenght | MMP-2 | K i app ≤ 9 pM | ? | [35] |
full-lenght | MMP-2 | IC50 3 nM | ? | [55] |
full-lenght | cdMMP-31 | K i 1.24 nM | ? | [57] |
full-lenght | MMP-3 | IC50 45 nM | ? | [55] |
full-lenght | MMP-3 | K i 1.51 nM | ? | [57] |
full-lenght | MMP-7 | IC50 8 nM | ? | [55] |
N-TIMP-4 | cdMMP-81 | K i 9.7 nM | Ser2 | [32] |
N-TIMP-4 | cdMMP-91 | K i 14.5 nM | Ser2 | [32] |
full-lenght | MMP-9 | IC50 83 nM | ? | [55] |
full-lenght | MMP-26 | IC50 0.4 nM | ? | [56] |
N-TIMP-4 | mbMT1-MMP3 | K i app 1.0 nM | ? | [33] |
full-lenght | sMT1-MMP3 | K i app 0.1 nM | ? | [35] |
N-TIMP-4 | ADAM-17/TACE | Ki 8.68 nM | ? | [65] |
full-lenght | ADAM-17/TACE | Ki 180 nM | ? | [65] |
full-lenght | cdADAM331 | Ki 220 nM | ? | [62] |