Classification | Compound | Structural formula | Compound | Structural formula |
---|---|---|---|---|
Pan-PI3K inhibitors | Pictilisib (GDC-0941) |
![]() | Copanlisib (BAY 80–6946) |
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Taselisib (GDC-0032) |
![]() | Sonolisib (PX-866) |
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Buparlisib (BKM120) |
![]() | ZSTK474 |
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Pilaralisib (XL147, SAR245408) |
![]() | AMG 511 |
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Isoform-selective inhibitors | Alpelisib (BYL719) |
![]() | CH5132799 |
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Idelalisib (CAL-101, GS-1101) |
![]() | AS-605240 |
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AMG319 |
![]() | MLN1117 (INK1117) |
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AZD6482 |
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Dual PI3K/mTOR inhibitors | Dactolisib (NVP-BEZ235) |
![]() | GDC-0084 (RG7666) |
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NVP-BGT226 |
![]() | VS-5584 (SB2343) |
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Omipalisib (GSK2126458, GSK458) |
![]() | PF-04691502 |
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GSK1059615 |
![]() | Gedatolisib (PF-05212384, PKI-587) |
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Voxtalisib (XL765, SAR245409) |
![]() | PQR309 |
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Apitolisib (GDC-0980) |
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